Tuesday, July 4, 2017

Safety of Gelatin Capsules vs HPMC Capsules

The PHD Chamber of Commerce & Industry ( PHDCCI) has submitted a representation to the Expert Committee headed by Dr. C. K. Kokate, Chairman, Expert Committee, Directorate General of Health Services, (DGHS), Ministry of Health and Family Welfare, Govt of India, in regard to the replacement of Gelatin Capsules with Cellulose Capsules as also the safety and vegetarian or non vegetarian aspects concerning Gelatine capsules versus HPMC capsules.

It may be noted that the DGHS vide notice dated June 02, 2017, had sought views of various stakeholders to address all the technical issues pertaining to replacement of gelatin capsules with cellulose based capsules for encapsulation of drugs.

The notice states that “A proposal has been received to replace gelatin capsules with cellulose based capsules which are of plant origin and are safe for use as compared to animal based gelatin capsules”.

Ministry of Health and Family Welfare vide order dated 20.03.2017 has constituted an Expert Committee to address all the technical issues pertaining to replacement of gelatin capsules with  cellulose based capsules for encapsulation of drugs.

The Committee has desired that views of stakeholders including manufacturers/marketers of HPMC capsules as well as NGOs who are working in this area or involved in this subject may also be obtained so that a considered view can be taken in the matter.  In order to examine the pros and cons of the proposal, suggestions/comments are invited from the Stakeholder/NGOs/Consumers within 21 days.

“In the meanwhile, soft gelatine capsules have been given a go-ahead, therefore there is no prima facie issue with the raw material and hence the replacement of the hard gelatine capsules being non-vegetarian is totally misplaced and uncalled for”, said Vivek Seigell, Director, PHD Chamber of Commerce & Industry said that the PHDCCI,

In this connection, at a meeting of the Technical Advisory Board (DTAB) of the CDSCO (the apex body to decide on technical issues) on May 13, 2016, a proposal to label cellulose based capsules with a green dot to indicate its vegetarian origin was considered. The DTAB turned down the proposal for the required amendment of the Drugs & Cosmetics Act on the basis that unlike in the case of food items, the choice of drugs is not that of the consumer (the patient) and is based on the prescription of the doctor where considerations of vegetarian origin or animal origin has no relevance. DTAB also recorded its observation that HPMC capsules are made from a semi synthetic chemical and hence cannot be considered of vegetarian origin.

The Supreme Court, in its order dated March 07, 2013, Case No. 641, had ordered that there is no need for non-veg or veg labels on drugs or cosmetics and hence even the red dots which are printed on non-veg products was not implemented for medicines.

According to Vivek Seigell, Director, PHD Chamber of Commerce & Industry, Gelatine Capsules are consumed by people at large as carriers of important medicines used to cure many terminal and lifestyle diseases. The consumption of medicine is more curative than out of personal choice. Looking at basic fundamental, it is not prudent to enter the Vegetarian and Non-Vegetarian debate in this matter. It may further be noted, that Gelatine used in the manufacture of empty capsules are derived from an extraction process wherein no animals are harmed or killed for this specific purpose. Only the left over bones having hydroxide and collagen, which is a protein widely found in animal bones (and is not more than 2% of the total value of the dead animal) is extracted through sophisticated machineries in WHO GMP approved extraction and manufacturing plants. Accordingly it is misplaced to have any notion that Gelatine Capsules are non-vegetarian in origin.

Gelatine capsules are totally safe for human consumption. WHO as per evidence certifies Empty Hard Gelatine Capsules for its total safety for Human Beings. And so do the Pharmacopoeia of USA, Japan,  European Union, United Kingdom, Australia and India.

When a scientific body of the Government of India, the Indian Pharmacopoeia Commission, publishes a monograph on gelatine and empty gelatine capsules how can it then be unsafe?  Presumably, the ultimate test of safety of a product is if it conforms to the specifications given in a pharmacopoeias, Several other pharmacopoeias around the world, including the British Pharmacopoeia, the United States Pharmacopoeia, and the Japanese Pharmacopoeia have confirmed its safety.

Inspite of the repeated requests Professor Kokate’s committee has not yet replied to stakeholders as to why gelatine capsules are less safe than HPMC (cellulose) capsules and what is the scientific and technical evidence for the same, if any.

“Across the globe over 95% of capsule formulations are gelatin capsules and even among the rest 5%, HPMC is primarily used for nutraceutical formulations. In India only around 2% capsules are HPMC based and almost all of them are nutraceuticals”, said Vivek Seigell. He further added that no cellulose capsules are used for products such as antibiotics, oncology, anti-infectious, painkiller and other medicinal categories. Nor have any tests been carried out by the DCGI in India whether such medicinal products would maintain their stability, bio-availability, bio-equivalence and other properties if filled in Cellulose capsules.

Technically speaking:

·        Pharmacokinetics and Pharmacodynamics properties of the drug has to be tested before it is put in to the market if the drug is encapsulated in Cellulose Capsules

·        Bioequivalence study for each drug would have to be carried out also

·        HPMC capsules are not suitable especially if the medicine has Potassium ions.  Similarly for a few of the drugs, Cellulose capsules were better than Gelatine capsules

·        At the same time a study of end of shelf life performance for cellulose based capsules needs to be conducted and, hence, the issue of replace of Gelatine should not be taken hastily


·        The time taken for the above tests of bioequivalence of thousands of drugs and combinations and Pharmacokinetics and Pharmacodynamics properties will take several years followed by the long process of approval from the drug authorities and any such move could mean devoiding the 1.2 billion people of this country of basic medical and health services for that many number of years.

 Following are the pointwise clarifications detailing the Myths and the Reality:

MYTH -1
HPMC CAPSULES ARE USED EXTENSIVELY IN MANY COUNTRIES

Reality
Over 95% of capsule formulations are  gelatin capsules and even among the rest 5%, HPMC is primarily used for nutraceutical formulations the World over . In  India only around 2% capsules are HPMC based and almost all of them are nutraceuticals.

MYTH -2
HPMC IS SAFER THAN GELATIN

Reality
Gelatin has been used for hard and soft capsules over the last 100 years and so far there has been practically  no reports of severe or even moderate adverse effects. On the other hand HPMC for Hard Capsules are of recent origin. Unlike in the case of production of Gelatin, HPMC manufacture involves use of reagents and chemicals, some of which are potential carcinogens,  in a multi step process..  The track record of HPMC use is just a decade or even less and therefore it is difficult to predict safety over time.

MYTH -3
HPMC OF THE RIGHT GRADE IS READILY AVAILABLE

Reality
The limited use of HPMC in India is dependent on imports (mostly from China) and it is not clear whether new generation HPMC, recommended for capsules is readily available and if they are, at what prices.

MYTH-4
REPLACEMENT OF GELATIN BY HPMC DOES NOT REQUIRE NEW REGULATORY APPROVALS

Reality
Any change of formulation and introduction of a new material or excipient is considered a New Drug under Schedule Y of the D&C Act. That means that every replaced formulation (with HPMC) of every API needs to be validated for safety, efficacy and pharmacokinetic parameters of dissolution, disintegration, release and  stability  through fresh pre clinical and/or clinical investigations. In fact if all hard gelatin capsules in the market ( close to 20,000 packs) are to be replaced, it will take several years to get them tested and approved and costs would be enormous  and that too at a time when every one is attempting to reduce healthcare costs  to make it more affordable for the masses.

MYTH- 5
CHANGE OVER TO HPMC WILL NOT ADD TO HIGHER COSTS OF THE CAPSULE FORMULATIONS

Reality
At present prices of HPMC , it is estimated that the costs  of production of HPMC capsules will be considerably  higher and so too prices. The new generation HPMC which is preferred for use in capsules is still patent protected and hence patent holders will have monopoly on prices.

MYTH – 6
ANIMALS ARE SLAUGHTERED FOR RAW MATERIAL (BONES, HIDES, FISH SCALES ETC. ) TO MANUFACTURE GELATIN

Reality
Raw materials used are waste products  of animals and animal derived foods, which  are environmentally unsafe and difficult to dispose off . Converting them to Gelatin and derived products adds value to waste material and offers solution to waste disposal issues. No animal is slaughtered for manufacture of Ossein, Gelatin and derived products

MYTH – 7
HPMC IS PLANT BASED AND THEREFORE NATURAL

Reality
While HPMC is based on Cellulose to start with, it undergoes chemical reactions involving building of new covalent linkages and hence is a chemical by definition and not a natural material

MYTH – 8
PRESENT PLANT AND MACHINERY CAN BE UTILIZED FOR MANUFACTURE OF HPMC CAPSULES

Reality
The process being different, considerable modification and fresh investments in new machinery would be required to produce HPMC capsules  

With the stoppage of Gelatine Capsules, both Cellulose capsules and Cellulose raw material will have to be imported at huge foreign exchange cost mainly from China, there by further increasing our dependence beyond the APIs which itself is quite precarious.  Additionally the capacity to supply HPMC capsules simply does not exist from overseas manufactures.

Vivek Seigell also pointed out that if it is an issue of non-vegetarian versus vegetarian capsules, then it should be noted that there has never been a bias against non-vegetarian sources in the manufacture of medicines. Products from non-vegetarian sources are currently widely used in many segments of pharmaceutical industry.

Gelatine is used in Blood plasma substitutes, Haemostatic sponges, Surgical implants, Hydrocolloidal dressings, Collagen for skin cream and Dietary supplements, certain food colours, vaccines, apart from auxiliary treatment for degenerative arthritic diseases and many other products, including a large number of food products.


95% of the Gelatine manufactured in India is produced by the PHDCCI Association members.  

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